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  Synthesis and Evaluation of¹¹ C-Labeled Triazolones as Probes for Imaging Fatty Acid Synthase Expression by Positron Emission Tomography

  Kelly, J. M., Jeitner, T. M., Waterhouse, N. N., Qu, W., Linstad, E. J., Samani, B., Williams, C., Nikolopoulou, A., Amor-Coarasa, A., Dimagno, S. G. & Babich, J. W., Mar 1 2022, In: Molecules. 27, 5, 1552.

  Research output: Contribution to journal › Article › peer-review

  Open Access

• Synthesis and evaluation of an acyl-chain unsaturated analog of the Th2 biasing, immunostimulatory glycolipid, OCH

  Velmourougane, G., Raju, R., Bricard, G., Im, J. S., Besra, G. S., Porcelli, S. A. & Howell, A. R., Jul 1 2009, In: Bioorganic and Medicinal Chemistry Letters. 19, 13, p. 3386-3388 3 p.

  Research output: Contribution to journal › Article › peer-review
  16 Scopus citations

• Synthesis and evaluation of antiproliferative activity of a geldanamycin-Herceptin(TM) immunoconjugate

  Mandler, R., Dadachova, E., Brechbiel, J. K., Waldmann, T. A. & Brechbiel, M. W., May 15 2000, In: Bioorganic and Medicinal Chemistry Letters. 10, 10, p. 1025-1028 4 p.

  Research output: Contribution to journal › Article › peer-review
  16 Scopus citations

• Synthesis and evaluation of new 4-phospho-D-erythronic acid derivatives as competitive inhibitors of spinach ribose-5-phosphate isomerase

  Burgos, E. & Salmon, L., Jan 19 2004, In: Tetrahedron Letters. 45, 4, p. 753-756 4 p.

  Research output: Contribution to journal › Article › peer-review
  11 Scopus citations

• Synthesis and evaluation of new antagonists of bacterial quorum sensing in Vibrio harveyi

  Peng, H., Cheng, Y., Ni, N., Li, M., Choudhary, G., Chou, H. T., Lu, C. D., Tai, P. C. & Wang, B., Sep 4 2009, In: ChemMedChem. 4, 9, p. 1457-1468 12 p.

  Research output: Contribution to journal › Article › peer-review
  46 Scopus citations

• Synthesis and evaluation of sphinganine analogues of KRN7000 and OCH

  Ndonye, R. M., Izmirian, D. P., Dunn, M. F., Yu, K. O. A., Porcelli, S. A., Khurana, A., Kronenberg, M., Richardson, S. K. & Howell, A. R., Dec 9 2005, In: Journal of Organic Chemistry. 70, 25, p. 10260-10270 11 p.

  Research output: Contribution to journal › Article › peer-review
  87 Scopus citations

• Synthesis and in vitro antimycobacterial activity of B-ring modified diaryl ether InhA inhibitors

  am Ende, C. W., Knudson, S. E., Liu, N., Childs, J., Sullivan, T. J., Boyne, M., Xu, H., Gegina, Y., Knudson, D. L., Johnson, F., Peloquin, C. A., Slayden, R. A. & Tonge, P. J., May 15 2008, In: Bioorganic and Medicinal Chemistry Letters. 18, 10, p. 3029-3033 5 p.

  Research output: Contribution to journal › Article › peer-review
  76 Scopus citations

• Synthesis and kinetic evaluation of 4-deoxy-4-phosphonomethyl-D- erythronate, the first hydrolytically stable and potent competitive inhibitor of ribose-5-phosphate isomerase

  Burgos, E. & Salmon, L., Apr 19 2004, In: Tetrahedron Letters. 45, 17, p. 3465-3469 5 p.

  Research output: Contribution to journal › Article › peer-review
  8 Scopus citations

• Synthesis and NMR characterization of the trypanosomatid metabolite, N ¹,N⁸-bis(glutathionyl)spermidine disulphide (trypanothione disulphide)

  Henderson, G. B., Glushka, J., Cowburn, D. & Cerami, A., 1990, In: Journal of the Chemical Society, Perkin Transactions 1. 4, p. 911-914 4 p.

  Research output: Contribution to journal › Article › peer-review
  22 Scopus citations

• Synthesis and pharmacological activity of 1,3,6-trisubstituted-4-oxo-1,4- dihydroquinoline-2-carboxylic acids as selective ET_A antagonists

  Patel, H. J., Olgun, N., Lengyel, I., Reznik, S. & Stephani, R. A., Nov 15 2010, In: Bioorganic and Medicinal Chemistry Letters. 20, 22, p. 6840-6844 5 p.

  Research output: Contribution to journal › Article › peer-review
  8 Scopus citations

• Synthesis and pre-clinical evaluation of a new class of high-affinity ¹⁸F-labeled PSMA ligands for detection of prostate cancer by PET imaging

  Kelly, J., Amor-Coarasa, A., Nikolopoulou, A., Kim, D., Williams, C., Ponnala, S. & Babich, J. W., Apr 1 2017, In: European Journal of Nuclear Medicine and Molecular Imaging. 44, 4, p. 647-661 15 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access
  43 Scopus citations

• Synthesis and preliminary biological evaluation of MMP inhibitor radiotracers [¹¹C]methyl-halo-CGS 27023A analogs, new potential PET breast cancer imaging agents

  Zheng, Q. H., Fei, X., Liu, X., Wang, J. Q., Bin Sun, H., Mock, B. H., Lee Stone, K., Martinez, T. D., Miller, K. D., Sledge, G. W. & Hutchins, G. D., Oct 2002, In: Nuclear Medicine and Biology. 29, 7, p. 761-770 10 p.

  Research output: Contribution to journal › Article › peer-review
  83 Scopus citations

• Synthesis and processing of precursor polypeptides to murine mammary tumor virus structural proteins

  Racevskis, J. & Sarkar, N. H., 1978, In: Journal of virology. 25, 1, p. 374-383 10 p.

  Research output: Contribution to journal › Article › peer-review
  28 Scopus citations

• Synthesis and processing of viral proteins in Friend erythroleukemia cell lines

  Racevskis, J. & Koch, G., Jun 15 1978, In: Virology. 87, 2, p. 354-365 12 p.

  Research output: Contribution to journal › Article › peer-review
  20 Scopus citations

• Synthesis and properties of 7-hydroxymethotrexate polyglutamyl derivatives in Ehrlich ascites tumor cells in vitro

  Fabre, G., Fabre, I., Matherly, L. H., Cano, J. P. & Goldman, I. D., 1984, In: Journal of Biological Chemistry. 259, 8, p. 5066-5072 7 p.

  Research output: Contribution to journal › Article › peer-review
  50 Scopus citations

• Synthesis and SAR studies of 1,4-benzoxazine MenB inhibitors: Novel antibacterial agents against Mycobacterium tuberculosis

  Li, X., Liu, N., Zhang, H., Knudson, S. E., Slayden, R. A. & Tonge, P. J., Nov 1 2010, In: Bioorganic and Medicinal Chemistry Letters. 20, 21, p. 6306-6309 4 p.

  Research output: Contribution to journal › Article › peer-review
  87 Scopus citations

• Synthesis and screening of a small glycomimetic library for inhibitory activity on medically relevant galactoside-specific lectins in assays of increasing biorelevance

  André, S., Giguère, D., Dam, T. K., Brewer, F., Gabius, H. J. & Roy, R., Oct 1 2010, In: New Journal of Chemistry. 34, 10, p. 2229-2240 12 p.

  Research output: Contribution to journal › Article › peer-review
  40 Scopus citations

• Synthesis and secretion of a high molecular weight form of nerve growth factor by skeletal muscle cells in culture

  Murphy, R. A., Singer, R. H., Saide, J. D., Pantazis, N. J., Blanchard, M. H., Byron, K. S., Arnason, B. G. & Young, M., 1977, In: Unknown Journal. 74, 10, p. 4496-4500 5 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access
  49 Scopus citations

• Synthesis and Structural Characterization of Ricin Inhibitors Targeting Ribosome Binding Using Fragment-Based Methods and Structure-Based Design

  Li, X. P., Harijan, R. K., Cao, B., Kahn, J. N., Pierce, M., Tsymbal, A. M., Roberge, J. Y., Augeri, D. & Tumer, N. E., Oct 28 2021, In: Journal of Medicinal Chemistry. 64, 20, p. 15334-15348 15 p.

  Research output: Contribution to journal › Article › peer-review
  2 Scopus citations

• Synthesis and structure of [Bp^But,Pri]₂Co: A bis(pyrazolyl)hydroborato cobalt(II) complex with trans [Co⋯H-B] interactions

  Ghosh, P., Bonanno, J. B. & Parkin, G., Jan 1 1998, In: Journal of the Chemical Society - Dalton Transactions. 17, p. 2779-2781 3 p.

  Research output: Contribution to journal › Article › peer-review
  21 Scopus citations

• Synthesis of (Z)-3,7-anhydro-1,2-dideoxy-2-deuterio-d-gluco-oct-2-enitol, a prochiral substrate for probing the catalytic functioning of glucosylases

  Weiser, W., Lehmann, J., Brewer, C. F. & Hehre, E. J., Dec 1 1988, In: Carbohydrate Research. 183, 2, p. 287-299 13 p.

  Research output: Contribution to journal › Article › peer-review
  11 Scopus citations

• Synthesis of [¹¹C]palmitic acid for PET imaging using a single molecular sieve 13X cartridge for reagent trapping, radiolabeling and selective purification

  Amor-Coarasa, A., Kelly, J. M. & Babich, J. W., Aug 1 2015, In: Nuclear Medicine and Biology. 42, 8, p. 685-690 6 p.

  Research output: Contribution to journal › Article › peer-review
  6 Scopus citations

• Synthesis of 1‐¹³C and 3‐¹³C isotopic isomers of aspartic and glutamic acids

  Fotadar, U. & Cowburn, D., 1983, In: Journal of Labelled Compounds and Radiopharmaceuticals. 20, 8, p. 1003-1009 7 p.

  Research output: Contribution to journal › Article › peer-review
  2 Scopus citations

• Synthesis of 4-phenoxybenzamide adenine dinucleotide as NAD analogue with inhibitory activity against enoyl-ACP reductase (InhA) of Mycobacterium tuberculosis

  Bonnac, L., Gao, G. Y., Chen, L., Felczak, K., Bennett, E. M., Xu, H., Kim, T. S., Liu, N., Oh, H. W., Tonge, P. J. & Pankiewicz, K. W., Aug 15 2007, In: Bioorganic and Medicinal Chemistry Letters. 17, 16, p. 4588-4591 4 p.

  Research output: Contribution to journal › Article › peer-review
  17 Scopus citations

• Synthesis of 5-benzyl and 5-benzyloxybenzyl 2,2'-anhydroudridines and related nucleoside analogs as inhibitors of uridine phosphorylase

  Chu, S. H., Weng, Z. Y., Chen, Z. H., Rowe, E. C., Chu, E., Naguib, F. N. M., el Kouni, M. H., Cha, S. & Chu, M. Y., Jan 2 1988, In: Nucleosides and Nucleotides. 7, 1, p. 91-102 12 p.

  Research output: Contribution to journal › Article › peer-review
  19 Scopus citations

• Synthesis of 5-deoxy-5-phospho-D-ribonohydroxamic acid: A new competitive and selective inhibitor of type B ribose-5-phosphate isomerase from Mycobacterium tuberculosis

  Burgos, E., Roos, A. K., Mowbray, S. L. & Salmon, L., May 23 2005, In: Tetrahedron Letters. 46, 21, p. 3691-3694 4 p.

  Research output: Contribution to journal › Article › peer-review
  9 Scopus citations

• Synthesis of 5-halogeno-6-amino-2'-deoxyuridines and their analogs as potential inhibitors of thymidine phosphorylase

  Pan, B. C., Chen, Z. H., Chu, E., WangChu, M. Y. & Chu, S. H., 1998, In: Nucleosides and Nucleotides. 17, 12, p. 2367-2382 16 p.

  Research output: Contribution to journal › Article › peer-review
  11 Scopus citations

• Synthesis of 5′-methylthio coformycins: Specific inhibitors for malarial adenosine deaminase

  Tyler, P. C., Taylor, E. A., Fröhlich, R. F. G. & Schramm, V. L., May 30 2007, In: Journal of the American Chemical Society. 129, 21, p. 6872-6879 8 p.

  Research output: Contribution to journal › Article › peer-review
  51 Scopus citations

• Synthesis of a carboxyl-terminal (constant region) fragment of the immunoglobin light chain by a mouse myeloma cell line

  Kuehl, W. M. & Scharff, M. D., Nov 5 1974, In: Journal of Molecular Biology. 89, 3, p. 409-412,IN1,413-421

  Research output: Contribution to journal › Article › peer-review
  41 Scopus citations

• Synthesis of all stereoisomers of KRN7000, the CD1d-binding NKT cell ligand

  Park, J. J., Lee, J. H., Ghosh, S. C., Bricard, G., Venkataswamy, M. M., Porcelli, S. A. & Chung, S. K., Jul 15 2008, In: Bioorganic and Medicinal Chemistry Letters. 18, 14, p. 3906-3909 4 p.

  Research output: Contribution to journal › Article › peer-review
  37 Scopus citations

• Synthesis of aminobenzyltriethylenetetraaminohexaacetic acid: Conjugation of the chelator to protein by an alkylamine linkage

  Bhargava, K. K., Zhang, Z. Y., Palestro, C. J. & Acharya, S. A., 1999, In: Journal of Protein Chemistry. 18, 7, p. 761-770 10 p.

  Research output: Contribution to journal › Article › peer-review

• Synthesis of aminobenzyltriethylenetetraaminohexaacetic acid: Conjugation of the chelator to protein by an alkylamine linkage

  Bhargava, K. K., Zhang, Z. Y., Palestro, C. J. & Acharya, S. A., 1999, In: Journal of Protein Chemistry. 18, 7, p. 761-770 10 p.

  Research output: Contribution to journal › Article › peer-review
  1 Scopus citations

• Synthesis of aminomethyl and amino analogs of 5‐benzylacyclouridine and 5‐benzyloxybenzylacyclouridine

  Chu, S. H., Chen, Z. H., Weng, Z. Y., Rowe, E. C., Chu, E. & Chu, MY. W., 1987, In: Journal of Heterocyclic Chemistry. 24, 4, p. 989-995 7 p.

  Research output: Contribution to journal › Article › peer-review
  8 Scopus citations

• Synthesis of a new 8-spin-labeled analog of adenosine 5'-phosphate and its interaction with AMP nucleosidase.

  DeWolf, W. E. & Schramm, V. L., Jul 25 1979, In: Journal of Biological Chemistry. 254, 14, p. 6215-6217 3 p.

  Research output: Contribution to journal › Article › peer-review
  2 Scopus citations

• Synthesis of a Photoaffinity Analog of Taxol as an Approach To Identify the Taxol Binding Site on Microtubules

  Carboni, J. M., Farina, V., Rao, S., Hauck, S. I., Horwitz, S. B. & Ringel, I., Jan 1 1993, In: Journal of Medicinal Chemistry. 36, 4, p. 513-515 3 p.

  Research output: Contribution to journal › Article › peer-review
  28 Scopus citations

• Synthesis of arbitrary frequency domain transmitting pulses applicable to pulsed NMR instruments

  Temps, A. J. & Brewer, C. F., Feb 15 1984, In: Journal of Magnetic Resonance (1969). 56, 3, p. 355-372 18 p.

  Research output: Contribution to journal › Article › peer-review
  37 Scopus citations

• Synthesis of a transition state analogue inhibitor of purine nucleoside phosphorylase via the Mannich reaction

  Evans, G. B., Furneaux, R. H., Tyler, P. C. & Schramm, V. L., Oct 2 2003, In: Organic Letters. 5, 20, p. 3639-3640 2 p.

  Research output: Contribution to journal › Article › peer-review
  82 Scopus citations

• Synthesis of bis-Phosphate Iminoaltritol Enantiomers and Structural Characterization with Adenine Phosphoribosyltransferase

  Harris, L. D., Harijan, R. K., Ducati, R. G., Evans, G. B., Hirsch, B. M. & Schramm, V. L., Jan 19 2018, In: ACS Chemical Biology. 13, 1, p. 152-160 9 p.

  Research output: Contribution to journal › Article › peer-review
  2 Scopus citations

• Synthesis of enantiomerically pure (2S,3S)-5,5,5-trifluoroisoleucine and (2R,3S)-5,5,5-trifluoro-allo-isoleucine

  Erdbrink, H., Nyakatura, E. K., Huhmann, S., Gerling, U. I. M., Lentz, D., Koksch, B. & Czekelius, C., Oct 2 2013, In: Beilstein Journal of Organic Chemistry. 9, p. 2009-2014 6 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access
  15 Scopus citations

• Synthesis of excess light chains of gamma globulin by rabbit lymph node cells

  Shapiro, A. L., Scharff, M. D., Maizel, J. V. & Uhr, J. W., 1966, In: Nature. 211, 5046, p. 243-245 3 p.

  Research output: Contribution to journal › Article › peer-review
  71 Scopus citations

• Synthesis of fluorescent phosphatidylinositols using a novel inositol H- phosphonate

  Leung, L. W., Vilchèze, C. & Bittman, R., May 7 1998, In: Tetrahedron Letters. 39, 19, p. 2921-2924 4 p.

  Research output: Contribution to journal › Article › peer-review
  9 Scopus citations

• Synthesis of folate- pegylated polyester nanoparticles encapsulating ixabepilone for targeting folate receptor overexpressing breast cancer cells

  Siafaka, P., Betsiou, M., Tsolou, A., Angelou, E., Agianian, B., Koffa, M., Chaitidou, S., Karavas, E., Avgoustakis, K. & Bikiaris, D., Dec 1 2015, In: Journal of Materials Science: Materials in Medicine. 26, 12, p. 1-14 14 p., 275.

  Research output: Contribution to journal › Article › peer-review
  43 Scopus citations

• Synthesis of GABA_A receptor agonists and evaluation of their α-subunit selectivity and orientation in the GABA binding site

  Jansen, M., Rabe, H., Strehle, A., Dieler, S., Debus, F., Dannhardt, G., Akabas, M. H. & Lüddens, H., Aug 14 2008, In: Journal of Medicinal Chemistry. 51, 15, p. 4430-4448 19 p.

  Research output: Contribution to journal › Article › peer-review
  36 Scopus citations

• Synthesis of hemispheric itd tuning from the readout of a neural map: Commonalities of proposed coding schemes in birds and mammals

  Pena, J. L., Cazettes, F., Beckert, M. V. & Fischer, B. J., Nov 13 2019, In: Journal of Neuroscience. 39, 46, p. 9053-9061 9 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access
  4 Scopus citations

• Synthesis of high molecular weight polyoxyethylene with a quaternary catalyst and study of its conductive blends with poly(2-vinyl pyridine)

  Xie, H. Q., Zhang, J. H., Cui, M. H. & Xie, D., Jul 15 2007, In: Journal of Applied Polymer Science. 105, 2, p. 562-569 8 p.

  Research output: Contribution to journal › Article › peer-review
  1 Scopus citations

• Synthesis of human plasminogen by the liver

  Raum, D., Marcus, D., Alper, C. A., Levey, R., Taylor, P. D. & Starzl, T. E., 1980, In: Science. 208, 4447, p. 1036-1037 2 p.

  Research output: Contribution to journal › Article › peer-review
  108 Scopus citations

• Synthesis of hyaluronic acid by human peritoneal mesothelial cells: Effect of cytokines and dialysate

  Breborowicz, A., Korybalska, K., Grzybowski, A., Wieczorowska-Tobis, K., Martis, L. & Oreopoulos, D. G., 1996, In: Peritoneal Dialysis International. 16, 4, p. 374-378 5 p.

  Research output: Contribution to journal › Article › peer-review
  25 Scopus citations

• Synthesis of immunoglobulin by substrate attached mouse myeloma cells

  Bargellesi, A., Damiani, G., Kuehl, W. M. & Scharff, M. D., Jun 1976, In: Journal of Cellular Physiology. 88, 2, p. 247-251 5 p.

  Research output: Contribution to journal › Article › peer-review
  6 Scopus citations

• Synthesis of melanin-like pigments by Sporothrix schenckii in vitro and during mammalian infection

  Morris-Jones, R., Youngchim, S., Gomez, B. L., Aisen, P., Hay, R. J., Nosanchuk, J. D., Casadevall, A. & Hamilton, A. J., Jul 1 2003, In: Infection and immunity. 71, 7, p. 4026-4033 8 p.

  Research output: Contribution to journal › Article › peer-review
  79 Scopus citations

• Synthesis of melanin pigment by Candida albicans in vitro and during infection

  Morris-Jones, R., Gomez, B. L., Diez, S., Uran, M., Morris-Jones, S. D., Casadevall, A., Nosanchuk, J. D. & Hamilton, A. J., Sep 2005, In: Infection and immunity. 73, 9, p. 6147-6150 4 p.

  Research output: Contribution to journal › Article › peer-review
  65 Scopus citations